Pharmakologie / Lesson
Parkinson-Medikamente
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- Zufuhr der DopaminvorstufeLevodopa + Decarboxylasehemmer: Carbidopa
- Dopamin- AgonistenBromocriptin D2 Ropinirol D2, D3 Pramipexol D3, D2 Apomorphin D1, D2 Rotigotin D3, D2, D1 Piribedil D2, D3
- MAO- B- HemmerSelegilin, Rasagilin
- COMT- HemmerEntacapon
- ParasympatholytikaBiperiden, Bornaprin, Trihexlphenidyl Hemmung exzitatorischer cholinerger Neurone → Acetylcholinspiegel↓
- NDMA-AntagonistenAmantadin, Memantin -> Hemmung glutamaterger Überreaktion
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