USMLE (Fach) / Pharmacology - Renal (Lektion)
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Losartan, candesartan, valsartan
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Selectively block binding of angiotensin II to AT1 receptor. Effects similar to ACE inhibitors, but ARBs do not increase bradykinin.
Use:- Hypertension- HF- Proteinuria- Chronic kidney disease (eg, diabetic nephropathy) with intolerance to ACE inhibitors (eg, cough, angioedema)
Adverse effects:- Hyperkalemia- ↓ GFR- Hypotension- Teratogen
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